Back to targets

Target detail

ACTR3

actin related protein 3

Data: Live structured evidence (Supabase)

Marker index metadata

Foundation row from public.targets — full Open Targets / ChEMBL preload remains a future operator job (Phase 8H+).

Display name: actin related protein 3

Aliases: ACTR3, actin related protein 3

Type / organism: protein_coding · Homo sapiens

Source: opentargets · ENSG00000115091

Index freshness: last_synced_at 2026-05-15T18:28:38.362+00:00 · updated 2026-05-15T18:28:38.813144+00:00

Limitations & build flags

  • Read-only structured navigator
  • No clinical outcome benefit inferred
  • Trial presence does not imply success
  • Drug identity may require normalization
  • Terminated/withdrawn trials must remain visible
Target index (foundation)

This symbol is listed in public.targets (operator seed or future preload). Connector-backed sections below may still show empty states until ChEMBL / Open Targets / ClinicalTrials.gov mirror rows exist for this marker.

Live structured evidence · sources

Connectors represented in loaded rows for ACTR3. Empty groups mean no matching rows — not a claim about biology or clinical use.

  • Open TargetsLive when indexed

    Disease–target evidence rows when operators run enrich:opentargets (GraphQL from trusted scripts only).

  • ChEMBLLive when indexed

    Drug–target and related enrichment rows when operators run enrich:chembl (server/CLI only).

  • CANTI signal builderLive when indexed

    Deterministic repurposing-signal rows produced by the in-repo signal builder when operators run the build pipeline.

Open Targets · disease–target evidence

Rows from disease_target_evidence for this symbol.

glioblastoma

literature · opentargets

ChEMBL · linked drugs (drug_targets)

Drug records tied via drug_targets — mechanistic linkage only.

Y-39983

chembl571948

Open drug

TAK-733

chembl1615025

Open drug

PELITINIB

chembl607707

Open drug

OSI-027

chembl3120215

Open drug

TUCATINIB

chembl3989868

Open drug

SNS-314

chembl482767

Open drug

VX-702

chembl1090090

Open drug

AMG-208

chembl496102

Open drug

TOVORAFENIB

chembl3348923

Open drug

PAZOPANIB

chembl477772

Open drug

ENCORAFENIB

chembl3301612

Open drug

REGORAFENIB

chembl1946170

Open drug

AMUVATINIB

chembl2103851

Open drug

SORAFENIB

chembl1336

Open drug

ULIXERTINIB

chembl3590106

Open drug

CHEMBL4129274

chembl4129274

Open drug

BMS-754807

chembl575448

Open drug

RABUSERTIB

chembl3039517

Open drug

VANDETANIB

chembl24828

Open drug

CRIZOTINIB

chembl601719

Open drug

TIRBANIBULIN

chembl571546

Open drug

PACRITINIB

chembl2035187

Open drug

FGFR INHIBITOR DEBIO 1347

chembl3907479

Open drug

GALUNISERTIB

chembl2364611

Open drug

AZD-6482

chembl2165191

Open drug

ENZASTAURIN

chembl300138

Open drug

AFATINIB

chembl1173655

Open drug

COBIMETINIB

chembl2146883

Open drug

XL-019

chembl3545328

Open drug

AZD-4547

chembl3184679

Open drug

MK-5108

chembl3600873

Open drug

AZD-8186

chembl3408248

Open drug

HMN-214

chembl3991927

Open drug

TAK-593

chembl2180604

Open drug

TIVOZANIB

chembl1289494

Open drug

FOSTAMATINIB

chembl2103830

Open drug

FEDRATINIB

chembl1287853

Open drug

AZD-5438

chembl488436

Open drug

PONATINIB

chembl1171837

Open drug

VEMURAFENIB

chembl1229517

Open drug

GOLVATINIB

chembl3039525

Open drug

CYC-116

chembl482967

Open drug

BUPARLISIB

chembl2017974

Open drug

DANUSERTIB

chembl402548

Open drug

SARACATINIB

chembl217092

Open drug

MK-2206

chembl1079175

Open drug

BGT-226 FREE BASE

chembl3218578

Open drug

LESTAURTINIB

chembl603469

Open drug

AMG-900

chembl2140408

Open drug

BOSUTINIB

chembl288441

Open drug

PICTILISIB

chembl521851

Open drug

CHEMBL2030402

chembl2030402

Open drug

NILOTINIB

chembl255863

Open drug

MOTESANIB

chembl572881

Open drug

TELATINIB

chembl2079588

Open drug

DECERNOTINIB

chembl3039513

Open drug

ENMD-2076

chembl482968

Open drug

OSI-632

chembl253969

Open drug

CHEMBL5653589

chembl5653589

Open drug

AV-412 FREE BASE

chembl2138625

Open drug

CHEMBL4084193

chembl4084193

Open drug

CHEMBL3991934

chembl3991934

Open drug

ROCILETINIB

chembl3545308

Open drug

PALBOCICLIB

chembl189963

Open drug

RUBOXISTAURIN

chembl91829

Open drug

GSK-461364

chembl1908394

Open drug

TG100-801

chembl403989

Open drug

SAR-407899 FREE BASE

chembl1667969

Open drug

OSIMERTINIB

chembl3353410

Open drug

CHEMBL3688339

chembl3688339

Open drug

CHEMBL3218575

chembl3218575

Open drug

TEMSIROLIMUS

chembl1201182

Open drug

LINIFANIB

chembl223360

Open drug

CHEMBL400402

chembl400402

Open drug

PF-04691502

chembl1234354

Open drug

SILMITASERTIB

chembl1230165

Open drug

SU-014813

chembl1721885

Open drug

LENVATINIB

chembl1289601

Open drug

IDELALISIB

chembl2216870

Open drug

CHEMBL3991935

chembl3991935

Open drug

BRIVANIB

chembl377300

Open drug

KW-2449

chembl1908397

Open drug

ENTRECTINIB

chembl1983268

Open drug

CUDC-101

chembl598797

Open drug

PF-03814735

chembl4289017

Open drug

SONOLISIB

chembl411907

Open drug

SELUMETINIB

chembl1614701

Open drug

MK-2461

chembl1822792

Open drug

DEFACTINIB

chembl3137331

Open drug

AC-480

chembl1645462

Open drug

CERITINIB

chembl2403108

Open drug

CHEMBL2376648

chembl2376648

Open drug

NMS-1286937

chembl1094408

Open drug

AFURESERTIB

chembl2219422

Open drug

RGB-286638

chembl3545083

Open drug

MERESTINIB

chembl3545307

Open drug

BI-2536

chembl513909

Open drug

AT-7519

chembl445813

Open drug

AZD-8055

chembl1801204

Open drug

MIDOSTAURIN

chembl608533

Open drug

SGI-1776

chembl1952329

Open drug

UCN-01

chembl574737

Open drug

CC-401

chembl1614713

Open drug

TANZISERTIB

chembl1950289

Open drug

RO-4987655

chembl1614766

Open drug

NINTEDANIB

chembl502835

Open drug

GSK-1070916

chembl1090479

Open drug

TAK-285

chembl1614725

Open drug

SUNITINIB

chembl535

Open drug

LINSITINIB

chembl1091644

Open drug

AT-9283

chembl495727

Open drug

MUBRITINIB

chembl1614707

Open drug

PERIFOSINE

chembl372764

Open drug

PF-03758309

chembl3128043

Open drug

IBRUTINIB

chembl1873475

Open drug

IMD-0354

chembl536151

Open drug

PIMASERTIB

chembl2107832

Open drug

RAF-265

chembl558752

Open drug

MK-8033

chembl2323775

Open drug

DASATINIB

chembl5416410

Open drug

DEFOSBARASERTIB

chembl215152

Open drug

LUCITANIB

chembl2220486

Open drug

CHEMBL3991933

chembl3991933

Open drug

TAK-901

chembl3544932

Open drug

CP-724714

chembl483321

Open drug

CHEMBL2048872

chembl2048872

Open drug

MIRDAMETINIB

chembl507361

Open drug

ALVOCIDIB

chembl428690

Open drug

BINIMETINIB

chembl3187723

Open drug

AEE-788

chembl587723

Open drug

MLN-8054

chembl259084

Open drug

BARICITINIB

chembl2105759

Open drug

BMS-911543

chembl3545215

Open drug

SOTRASTAURIN

chembl565612

Open drug

BMS-387032

chembl296468

Open drug

PHA-793887

chembl1230607

Open drug

GLESATINIB

chembl3989914

Open drug

AT-13148

chembl3544960

Open drug

AZD-8330

chembl3182621

Open drug

ICOTINIB

chembl2087361

Open drug

ERLOTINIB

chembl553

Open drug

DACOMITINIB ANHYDROUS

chembl2110732

Open drug

CABOZANTINIB

chembl2105717

Open drug

CAPMATINIB

chembl3188267

Open drug

K-252A

chembl281948

Open drug

GSK-1059615

chembl3544966

Open drug

ALPELISIB

chembl2396661

Open drug

UPROSERTIB

chembl3137336

Open drug

GILTERITINIB

chembl3301622

Open drug

DABRAFENIB

chembl2028663

Open drug

CEDIRANIB

chembl491473

Open drug

GSK-690693

chembl494089

Open drug

QUIZARTINIB

chembl576982

Open drug

WHI-P131

chembl405130

Open drug

ALECTINIB

chembl1738797

Open drug

TEPOTINIB

chembl3402762

Open drug

TRAMETINIB

chembl2103875

Open drug

TIDEGLUSIB

chembl3545157

Open drug

VOXTALISIB

chembl3545366

Open drug

PEXMETINIB

chembl3991932

Open drug

CRENOLANIB

chembl2105728

Open drug

RAVOXERTINIB

chembl3544964

Open drug

AZD-7762

chembl2041933

Open drug

DOVITINIB

chembl522892

Open drug

AZD-1480

chembl1231124

Open drug

R-406

chembl475251

Open drug

AXL-1717

chembl283120

Open drug

COPANLISIB

chembl3218576

Open drug

REBASTINIB

chembl1738757

Open drug

RIDAFOROLIMUS

chembl2103839

Open drug

RIGOSERTIB

chembl1241855

Open drug

LAPATINIB

chembl554

Open drug

MOMELOTINIB

chembl1078178

Open drug

PF-00562271

chembl1084546

Open drug

EVEROLIMUS

chembl1908360

Open drug

DACTOLISIB

chembl1879463

Open drug

Cerdulatinib Hydrochloride

chembl3991929

Open drug

GEDATOLISIB

chembl592445

Open drug

ORANTINIB

chembl274654

Open drug

VATALANIB

chembl101253

Open drug

HYDROXYFASUDIL

chembl1233300

Open drug

BARASERTIB

chembl415049

Open drug

APITOLISIB

chembl1922094

Open drug

AEW-541

chembl551064

Open drug

SCH-900776

chembl2386889

Open drug

CHEMBL3699142

chembl3699142

Open drug

PEXIDARTINIB

chembl3813873

Open drug

LOSMAPIMOD

chembl1088752

Open drug

FILGOTINIB

chembl3301607

Open drug

RIVOCERANIB

chembl3186534

Open drug

CANERTINIB

chembl31965

Open drug

TANDUTINIB

chembl124660

Open drug

GEFITINIB

chembl939

Open drug

DINACICLIB

chembl2103840

Open drug

TESEVATINIB

chembl3544983

Open drug

JNJ-38877605

chembl2133806

Open drug

TIVANTINIB

chembl2103882

Open drug

TOFACITINIB

chembl221959

Open drug

ADAVOSERTIB

chembl1976040

Open drug

XL-228

chembl3545085

Open drug
repoDB-style · approved-elsewhere discussion candidates

disease_drug_evidence rows on linked drugs whose evidence_type suggests approved-elsewhere discussion context.

No matching rows

Import repoDB-compatible disease–drug evidence or add structured rows to surface discussion candidates here.

ClinicalTrials.gov · trial-matched options

Mirror rows whose text fields mention this symbol — registry context only.

No matching live evidence found

Populate clinical_trials via the registry enrichment flow; this panel matches the symbol token in titles, conditions, or interventions.

CANTI signal builder · target-linked research signals

Repurposing signal rows for drugs linked to this target via drug_targets.

Repurposing research signal · BOSUTINIB · v0.1

Deterministic research signal for BOSUTINIB. Aggregate template score 55 (not a clinical endpoint). Contributing canonical sources observed in this rollup: chembl, opentargets. No failed-repoDB or terminated-trial penalty lines fired for this rollup. Missing relative to the Phase 8A template: glioma/brain-tumor–scoped ClinicalTrials.gov disease–drug evidence; repoDB-style disease–drug labels. This row requires clinical/research review before any operational use — not care-planning guidance, dose planning, or outcome-benefit claims.

Open signals hub

Repurposing research signal · AT-9283 · v0.1

Deterministic research signal for AT-9283. Aggregate template score 55 (not a clinical endpoint). Contributing canonical sources observed in this rollup: chembl, opentargets. No failed-repoDB or terminated-trial penalty lines fired for this rollup. Missing relative to the Phase 8A template: glioma/brain-tumor–scoped ClinicalTrials.gov disease–drug evidence; repoDB-style disease–drug labels. This row requires clinical/research review before any operational use — not care-planning guidance, dose planning, or outcome-benefit claims.

Open signals hub

Repurposing research signal · ALVOCIDIB · v0.1

Deterministic research signal for ALVOCIDIB. Aggregate template score 55 (not a clinical endpoint). Contributing canonical sources observed in this rollup: chembl, opentargets. No failed-repoDB or terminated-trial penalty lines fired for this rollup. Missing relative to the Phase 8A template: glioma/brain-tumor–scoped ClinicalTrials.gov disease–drug evidence; repoDB-style disease–drug labels. This row requires clinical/research review before any operational use — not care-planning guidance, dose planning, or outcome-benefit claims.

Open signals hub

Repurposing research signal · BMS-387032 · v0.1

Deterministic research signal for BMS-387032. Aggregate template score 55 (not a clinical endpoint). Contributing canonical sources observed in this rollup: chembl, opentargets. No failed-repoDB or terminated-trial penalty lines fired for this rollup. Missing relative to the Phase 8A template: glioma/brain-tumor–scoped ClinicalTrials.gov disease–drug evidence; repoDB-style disease–drug labels. This row requires clinical/research review before any operational use — not care-planning guidance, dose planning, or outcome-benefit claims.

Open signals hub

Repurposing research signal · CANERTINIB · v0.1

Deterministic research signal for CANERTINIB. Aggregate template score 55 (not a clinical endpoint). Contributing canonical sources observed in this rollup: chembl, opentargets. No failed-repoDB or terminated-trial penalty lines fired for this rollup. Missing relative to the Phase 8A template: glioma/brain-tumor–scoped ClinicalTrials.gov disease–drug evidence; repoDB-style disease–drug labels. This row requires clinical/research review before any operational use — not care-planning guidance, dose planning, or outcome-benefit claims.

Open signals hub

Repurposing research signal · CEP-32496 · v0.1

Deterministic research signal for CEP-32496. Aggregate template score 55 (not a clinical endpoint). Contributing canonical sources observed in this rollup: chembl, opentargets. No failed-repoDB or terminated-trial penalty lines fired for this rollup. Missing relative to the Phase 8A template: glioma/brain-tumor–scoped ClinicalTrials.gov disease–drug evidence; repoDB-style disease–drug labels. This row requires clinical/research review before any operational use — not care-planning guidance, dose planning, or outcome-benefit claims.

Open signals hub

Repurposing research signal · BAFETINIB · v0.1

Deterministic research signal for BAFETINIB. Aggregate template score 55 (not a clinical endpoint). Contributing canonical sources observed in this rollup: chembl, opentargets. No failed-repoDB or terminated-trial penalty lines fired for this rollup. Missing relative to the Phase 8A template: glioma/brain-tumor–scoped ClinicalTrials.gov disease–drug evidence; repoDB-style disease–drug labels. This row requires clinical/research review before any operational use — not care-planning guidance, dose planning, or outcome-benefit claims.

Open signals hub
Caution / negative-evidence rows

Structured rows with negative evidence_direction on disease–drug or signal tables.

No negative-direction rows

When structured evidence includes explicit negative direction fields, they surface here for oncology review.

Missing evidence · row counts by source string

No ClinicalTrials.gov mirror rows mention this symbol in titles, conditions, or interventions (within the loaded window).

  • chembl: 238
  • canti_signal_builder: 7
  • opentargets: 1
Summary row (aggregated list)

Structured evidence rows link this marker to cohort contexts when ingested — interpret as research context only.

Disease contexts

0

Linked drugs

0

Linked in dataset

0

Research signals

0

Evidence badges (illustrative)

Doctor-discussion candidate and related tags are descriptive only.

Appears in source landscapeLinked in datasetRequires oncology review
Linked research signals (list read)

Signals list: Live structured evidence (Supabase)

Repurposing research signal · ALVOCIDIB · v0.1

Deterministic research signal for ALVOCIDIB. Aggregate template score 55 (not a clinical endpoint). Contributing canonical sources observed in this rollup: chembl, opentargets. No failed-repoDB or terminated-trial penalty lines fired for this rollup. Missing relative to the Phase 8A template: glioma/brain-tumor–scoped ClinicalTrials.gov disease–drug evidence; repoDB-style disease–drug labels. This row requires clinical/research review before any operational use — not care-planning guidance, dose planning, or outcome-benefit claims.

View signals hub

Repurposing research signal · CEP-32496 · v0.1

Deterministic research signal for CEP-32496. Aggregate template score 55 (not a clinical endpoint). Contributing canonical sources observed in this rollup: chembl, opentargets. No failed-repoDB or terminated-trial penalty lines fired for this rollup. Missing relative to the Phase 8A template: glioma/brain-tumor–scoped ClinicalTrials.gov disease–drug evidence; repoDB-style disease–drug labels. This row requires clinical/research review before any operational use — not care-planning guidance, dose planning, or outcome-benefit claims.

View signals hub

Repurposing research signal · CANERTINIB · v0.1

Deterministic research signal for CANERTINIB. Aggregate template score 55 (not a clinical endpoint). Contributing canonical sources observed in this rollup: chembl, opentargets. No failed-repoDB or terminated-trial penalty lines fired for this rollup. Missing relative to the Phase 8A template: glioma/brain-tumor–scoped ClinicalTrials.gov disease–drug evidence; repoDB-style disease–drug labels. This row requires clinical/research review before any operational use — not care-planning guidance, dose planning, or outcome-benefit claims.

View signals hub

Repurposing research signal · BOSUTINIB · v0.1

Deterministic research signal for BOSUTINIB. Aggregate template score 55 (not a clinical endpoint). Contributing canonical sources observed in this rollup: chembl, opentargets. No failed-repoDB or terminated-trial penalty lines fired for this rollup. Missing relative to the Phase 8A template: glioma/brain-tumor–scoped ClinicalTrials.gov disease–drug evidence; repoDB-style disease–drug labels. This row requires clinical/research review before any operational use — not care-planning guidance, dose planning, or outcome-benefit claims.

View signals hub

Repurposing research signal · BMS-387032 · v0.1

Deterministic research signal for BMS-387032. Aggregate template score 55 (not a clinical endpoint). Contributing canonical sources observed in this rollup: chembl, opentargets. No failed-repoDB or terminated-trial penalty lines fired for this rollup. Missing relative to the Phase 8A template: glioma/brain-tumor–scoped ClinicalTrials.gov disease–drug evidence; repoDB-style disease–drug labels. This row requires clinical/research review before any operational use — not care-planning guidance, dose planning, or outcome-benefit claims.

View signals hub

Repurposing research signal · AT-9283 · v0.1

Deterministic research signal for AT-9283. Aggregate template score 55 (not a clinical endpoint). Contributing canonical sources observed in this rollup: chembl, opentargets. No failed-repoDB or terminated-trial penalty lines fired for this rollup. Missing relative to the Phase 8A template: glioma/brain-tumor–scoped ClinicalTrials.gov disease–drug evidence; repoDB-style disease–drug labels. This row requires clinical/research review before any operational use — not care-planning guidance, dose planning, or outcome-benefit claims.

View signals hub

Repurposing research signal · BAFETINIB · v0.1

Deterministic research signal for BAFETINIB. Aggregate template score 55 (not a clinical endpoint). Contributing canonical sources observed in this rollup: chembl, opentargets. No failed-repoDB or terminated-trial penalty lines fired for this rollup. Missing relative to the Phase 8A template: glioma/brain-tumor–scoped ClinicalTrials.gov disease–drug evidence; repoDB-style disease–drug labels. This row requires clinical/research review before any operational use — not care-planning guidance, dose planning, or outcome-benefit claims.

View signals hub